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Chemotherapy was potentiated by E7449 and solitary agent had important antitumor exercise in BRCA-deficient xenografts. Additionally, E7449 inhibited Wnt/β-catenin signaling in colon most cancers cell lines, likely via TNKS inhibition. In keeping with this risk, E7449 stabilized axin and TNKS proteins resulting in β-catenin de-stabilization and appreciably altered expression of https://mariokdulc.blogcudinti.com/29351634/the-2-minute-rule-for-apigenin

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